Cluster composition

Functions

CategoryNameIntersectionWithQueryPValueGenesInTermGenesInQueryGenesInTermInQueryID
GeneOntologyMolecularFunctiontranscription factor binding

TRERF1 CCNT2 SETD1A NCOR2 NCOA6 CRTC3 PTPRN EGR2 NFATC4 KDM5C SIN3A MED1 SPEN TOX2 HDAC7 TBX5

5.83e-087538216GO:0008134
GeneOntologyMolecularFunctionDNA-binding transcription factor binding

TRERF1 SETD1A NCOR2 NCOA6 CRTC3 EGR2 KDM5C SIN3A MED1 SPEN TOX2 HDAC7 TBX5

6.78e-075828213GO:0140297
GeneOntologyMolecularFunctionRNA polymerase II-specific DNA-binding transcription factor binding

TRERF1 SETD1A NCOR2 NCOA6 EGR2 KDM5C SIN3A MED1 SPEN TOX2 TBX5

1.07e-064178211GO:0061629
GeneOntologyMolecularFunctiontranscription coregulator activity

TRERF1 NCOR2 NCOA6 ZMIZ2 NFKBIZ SIN3A MED1 CBFA2T3 SPEN TOX2 HDAC7 TRIM52

3.03e-065628212GO:0003712
GeneOntologyMolecularFunctiontranscription corepressor activity

TRERF1 NCOR2 SIN3A MED1 CBFA2T3 SPEN HDAC7

4.36e-05229827GO:0003714
GeneOntologyMolecularFunctionperoxisome proliferator activated receptor binding

NCOA6 NFATC4 MED1

8.42e-0521823GO:0042975
GeneOntologyMolecularFunctionnuclear receptor coactivator activity

TRERF1 NCOA6 ZMIZ2 MED1

1.15e-0461824GO:0030374
GeneOntologyMolecularFunctionchromatin binding

CCNT2 NCOR2 NCOA6 ATF5 EGR2 GLI1 SIN3A MED1 CBFA2T3 TOX2 HDAC7

2.12e-047398211GO:0003682
GeneOntologyMolecularFunctionSUMO transferase activity

EGR2 ZMIZ2 HDAC7

4.32e-0436823GO:0019789
GeneOntologyMolecularFunctionhistone H3K4 monomethyltransferase activity

SETD1A SETD1B

4.59e-048822GO:0140945
GeneOntologyMolecularFunctionhistone H3K4 trimethyltransferase activity

SETD1A SETD1B

7.34e-0410822GO:0140999
GeneOntologyMolecularFunctionprotein-macromolecule adaptor activity

TRERF1 NCOR2 NCOA6 ZMIZ2 DVL2 NFKBIZ SIN3A MED1 CBFA2T3 SPEN TOX2 HDAC7 TRIM52

8.48e-0411608213GO:0030674
GeneOntologyMolecularFunctiontranscription coactivator binding

TRERF1 CCNT2 MED1

1.42e-0354823GO:0001223
GeneOntologyMolecularFunctionnuclear retinoic acid receptor binding

NCOR2 NCOA6 MED1

1.50e-0355823GO:0042974
GeneOntologyMolecularFunctiontranscription coactivator activity

TRERF1 NCOA6 ZMIZ2 MED1 TOX2 TRIM52

1.55e-03303826GO:0003713
GeneOntologyMolecularFunctionnuclear vitamin D receptor binding

NCOA6 MED1

2.44e-0318822GO:0042809
GeneOntologyMolecularFunctionnuclear glucocorticoid receptor binding

NCOR2 NCOA6

3.02e-0320822GO:0035259
GeneOntologyMolecularFunctionhistone H3K4 methyltransferase activity

SETD1A SETD1B

3.02e-0320822GO:0042800
GeneOntologyMolecularFunctionSUMO ligase activity

EGR2 ZMIZ2

3.02e-0320822GO:0061665
GeneOntologyMolecularFunctionprotein domain specific binding

WBP1 NCOA6 EGR2 WASF2 KHDRBS2 DVL2 IST1 NFKBIZ PLSCR3 MED1

3.05e-038758210GO:0019904
GeneOntologyBiologicalProcesspositive regulation of transcription by RNA polymerase II

TRERF1 ZNF462 CCNT2 NCOA6 CRTC3 ELL2 ATF5 PTPRN EGR2 NFATC4 GLI1 ZMIZ2 SOX30 DVL2 LRP6 NFKBIZ MED1 TOX2 CDON SP7 TBX5

4.68e-0813908021GO:0045944
GeneOntologyBiologicalProcessbrain development

ATP5PB SETD1A NCOR2 NCOA6 ATF5 EGR2 GLI1 USP9X LRP6 ROBO2 SIN3A MED1 CDON

2.46e-058598013GO:0007420
GeneOntologyBiologicalProcesshead development

ATP5PB SETD1A NCOR2 NCOA6 ATF5 EGR2 GLI1 USP9X LRP6 ROBO2 SIN3A MED1 CDON

4.95e-059198013GO:0060322
DomainN-SET

SETD1A SETD1B

1.86e-052812PF11764
DomainCOMPASS_Set1_N-SET

SETD1A SETD1B

1.86e-052812IPR024657
DomainN-SET

SETD1A SETD1B

1.86e-052812SM01291
DomainPost-SET_dom

SETD1A SETD1B

2.14e-0316812IPR003616
DomainPostSET

SETD1A SETD1B

2.14e-0316812SM00508
DomainPOST_SET

SETD1A SETD1B

2.14e-0316812PS50868
DomainPentatricopeptide_repeat

DTNB POLRMT

4.43e-0323812IPR002885
DomainSANT_dom

TRERF1 NCOR2

5.64e-0326812IPR017884
DomainSANT

TRERF1 NCOR2

6.53e-0328812PS51293
DomainPH

IQSEC2 ARHGEF9 OBSCN TRIOBP PLEKHA7

7.20e-03278815SM00233
DomainPH_DOMAIN

IQSEC2 ARHGEF9 OBSCN TRIOBP PLEKHA7

7.31e-03279815PS50003
DomainPH_domain

IQSEC2 ARHGEF9 OBSCN TRIOBP PLEKHA7

7.41e-03280815IPR001849
PathwayWP_HEDGEHOG_SIGNALING_WP47

GLI1 PTCH2 SIN3A

3.95e-0516603M39675
PathwayREACTOME_MITOCHONDRIAL_BIOGENESIS

ATP5PB NCOA6 CRTC3 POLRMT MED1

5.36e-0596605M26973
PathwayREACTOME_REGULATION_OF_LIPID_METABOLISM_BY_PPARALPHA

NCOR2 SIN3A MED1

5.72e-0518603MM15034
PathwayREACTOME_TRANSCRIPTIONAL_ACTIVATION_OF_MITOCHONDRIAL_BIOGENESIS

NCOA6 CRTC3 POLRMT MED1

8.60e-0555604M27145
PathwayWP_HEDGEHOG_SIGNALING_PATHWAY

GLI1 PTCH2 SIN3A

1.07e-0422603MM15924
PathwayREACTOME_CYTOPROTECTION_BY_HMOX1

NCOR2 NCOA6 SIN3A MED1

1.21e-0460604M41830
PathwayBIOCARTA_CARM_ER_PATHWAY

NCOR2 MED1 SPEN

1.78e-0426603M2499
PathwayREACTOME_GENE_EXPRESSION_TRANSCRIPTION

CCNT2 CASC3 SETD1A NCOR2 ELL2 SETD1B USP9X PIP4P1 POLRMT SIN3A MED1 HDAC7 TBX5

2.97e-0410226013MM15436
PathwayREACTOME_GLI_PROTEINS_BIND_PROMOTERS_OF_HH_RESPONSIVE_GENES_TO_PROMOTE_TRANSCRIPTION

GLI1 PTCH2

3.69e-047602M27501
PathwayREACTOME_TRANSCRIPTIONAL_REGULATION_OF_WHITE_ADIPOCYTE_DIFFERENTIATION

NCOR2 NCOA6 EGR2 MED1

4.44e-0484604M1008
PathwayKEGG_MEDICUS_REFERENCE_HEDGEHOG_SIGNALING_PATHWAY_PTCH_CORECEPTOR

PTCH2 CDON

6.29e-049602M47893
PathwayREACTOME_TRANSCRIPTIONAL_ACTIVITY_OF_SMAD2_SMAD3_SMAD4_HETEROTRIMER

CCNT2 NCOR2 USP9X

6.96e-0441603MM14876
PathwayREACTOME_FORMATION_OF_WDR5_CONTAINING_HISTONE_MODIFYING_COMPLEXES

SETD1A NCOA6 SETD1B

7.48e-0442603M48018
PathwayWP_HEDGEHOG_SIGNALING_WP4249

GLI1 PTCH2 CDON

8.01e-0443603M39706
PathwayREACTOME_RUNX1_REGULATES_GENES_INVOLVED_IN_MEGAKARYOCYTE_DIFFERENTIATION_AND_PLATELET_FUNCTION

SETD1A SETD1B SIN3A

8.57e-0444603MM15527
PathwayREACTOME_HEME_SIGNALING

NCOA6 CRTC3 MED1

1.18e-0349603M41832
PathwayREACTOME_ADIPOGENESIS

NCOR2 NCOA6 EGR2 MED1

1.22e-03110604M48259
PathwayREACTOME_TRANSCRIPTIONAL_ACTIVITY_OF_SMAD2_SMAD3_SMAD4_HETEROTRIMER

CCNT2 NCOR2 USP9X

1.32e-0351603M665
PathwayREACTOME_LOSS_OF_FUNCTION_OF_MECP2_IN_RETT_SYNDROME

NCOR2 SIN3A

1.35e-0313602M29766
PathwayREACTOME_GENERIC_TRANSCRIPTION_PATHWAY

CCNT2 SETD1A NCOR2 SETD1B USP9X PIP4P1 SIN3A MED1 HDAC7 TBX5

1.37e-037686010MM14851
PathwayREACTOME_CYTOPROTECTION_BY_HMOX1

NCOR2 SIN3A MED1

1.40e-0352603MM15684
PathwayKEGG_MEDICUS_REFERENCE_HEDGEHOG_SIGNALING_PATHWAY

GLI1 PTCH2

1.57e-0314602M47414
PathwayREACTOME_REGULATION_OF_LIPID_METABOLISM_BY_PPARALPHA

NCOR2 NCOA6 SIN3A MED1

1.59e-03118604M27316
PathwayKEGG_BASAL_CELL_CARCINOMA

GLI1 DVL2 PTCH2

1.64e-0355603M17807
PathwayREACTOME_RNA_POLYMERASE_II_TRANSCRIPTION

CCNT2 CASC3 SETD1A NCOR2 ELL2 SETD1B RBFOX3 USP9X PIP4P1 SIN3A MED1 HDAC7 SP7 TBX5

1.70e-0313876014M734
Pubmed

Proteome-scale mapping of binding sites in the unstructured regions of the human proteome.

TRERF1 WBP1 SETD1A NCOR2 NCOA6 CRTC3 ZNF469 ATF5 EGR2 NFATC4 BICRA ZMIZ2 PIP4P1 SIN3A SPEN PLEKHA7 VPS37B RNF11

9.07e-18430821835044719
Pubmed

Human transcription factor protein interaction networks.

TRERF1 ATP5PB ZNF462 PRR12 SETD1A NCOR2 NCOA6 GSE1 NFATC4 BICRA PRRC2C USP9X ZMIZ2 PIP4P1 LRP6 PROSER1 SIN3A NDUFA8 SPEN CCDC86 SP7

1.11e-111429822135140242
Pubmed

Interaction network of human early embryonic transcription factors.

TRERF1 ZNF462 PRR12 SETD1A NCOR2 NCOA6 GSE1 EGR2 BICRA ZMIZ2 PROSER1 SPEN

4.07e-11351821238297188
Pubmed

The Eyes Absent family members EYA4 and EYA1 promote PLK1 activation and successful mitosis through tyrosine dephosphorylation.

PRR12 NCOR2 GSE1 BICRA ZMIZ2 CCDC120 PROSER1 VPS37B

3.00e-0915282838360978
Pubmed

Control of developmentally primed erythroid genes by combinatorial co-repressor actions.

NCOR2 GSE1 SIN3A CBFA2T3 SPEN

8.76e-093082526593974
Pubmed

Large-scale characterization of HeLa cell nuclear phosphoproteins.

TRERF1 CCNT2 NCOR2 MYOF NCOA6 GSE1 KDM5C TJAP1 SIN3A MED1 SPEN CCDC86 HDAC7

3.23e-08774821315302935
Pubmed

Identification of the SOX2 Interactome by BioID Reveals EP300 as a Mediator of SOX2-dependent Squamous Differentiation and Lung Squamous Cell Carcinoma Growth.

PRR12 NCOR2 NCOA6 GSE1 MED1 SPEN

4.66e-088382628794006
Pubmed

Proteomic analyses reveal distinct chromatin-associated and soluble transcription factor complexes.

NCOR2 GSE1 NFATC4 PRRC2C GLI1 KDM5C WASF2 DVL2 POLRMT SIN3A CBFA2T3 SPEN CCDC86

1.05e-07857821325609649
Pubmed

Isolation of a novel histone deacetylase reveals that class I and class II deacetylases promote SMRT-mediated repression.

NCOR2 SIN3A HDAC7

1.26e-07582310640276
Pubmed

An inducible CRISPR/Cas9 screen identifies DTX2 as a transcriptional regulator of human telomerase.

PRR12 NCOR2 CRTC3 GSE1 TMEM209 CCDC120 PLEKHA7

2.43e-0718082735198878
Pubmed

Deficiency of Wdr60 and Wdr34 cause distinct neural tube malformation phenotypes in early embryos.

SETD1A GLI1 PTCH2 LRP6

4.12e-072682437228654
Pubmed

The transcriptional corepressor MTG16a contains a novel nucleolar targeting sequence deranged in t (16; 21)-positive myeloid malignancies.

NCOR2 SIN3A CBFA2T3

4.39e-07782312242670
Pubmed

A distinct Smoothened mutation causes severe cerebellar developmental defects and medulloblastoma in a novel transgenic mouse model.

RBFOX3 GLI1 PTCH2

7.01e-07882322869526
Pubmed

Agonist-specific Protein Interactomes of Glucocorticoid and Androgen Receptor as Revealed by Proximity Mapping.

NCOR2 NCOA6 GSE1 MED1 SPEN

1.19e-067882528611094
Pubmed

Comparative Application of BioID and TurboID for Protein-Proximity Biotinylation.

PRR12 NCOR2 NCOA6 CRTC3 GSE1 PRRC2C GLI1 TMEM209 POLRMT

1.35e-0645782932344865
Pubmed

A dual-activity topoisomerase complex regulates mRNA translation and turnover.

PRR12 SETD1A NCOR2 MYOF NCOA6 SETD1B BICRA GLI1 ZMIZ2 OBSCN POLRMT SPEN HDAC7

1.83e-061105821335748872
Pubmed

Spatiotemporal profile of postsynaptic interactomes integrates components of complex brain disorders.

TRERF1 ZNF462 CASC3 NCOR2 PRRC2C USP9X WASF2 IQSEC2 CNKSR3 DVL2 TRIOBP TJAP1

2.65e-06963821228671696
Pubmed

Lhx2 is a progenitor-intrinsic modulator of Sonic Hedgehog signaling during early retinal neurogenesis.

GLI1 PTCH2 CDON

2.74e-061282336459481
Pubmed

Wnt1 Lineage Specific Deletion of Gpr161 Results in Embryonic Midbrain Malformation and Failure of Craniofacial Skeletal Development.

GLI1 DVL2 LRP6

3.55e-061382334887903
Pubmed

Ptch2/Gas1 and Ptch1/Boc differentially regulate Hedgehog signalling in murine primordial germ cell migration.

GLI1 PTCH2 CDON

3.55e-061382332332736
Pubmed

Chemoproteomics profiling of HDAC inhibitors reveals selective targeting of HDAC complexes.

TRERF1 NCOR2 GSE1 SIN3A

3.97e-064582421258344
Pubmed

Comparative sequence and x-inactivation analyses of a domain of escape in human xp11.2 and the conserved segment in mouse.

KDM5C IQSEC2

5.49e-06282215197169
Pubmed

The H3K4 methyltransferase Setd1a is first required at the epiblast stage, whereas Setd1b becomes essential after gastrulation.

SETD1A SETD1B

5.49e-06282224550110
Pubmed

Myoferlin Regulates Wnt/β-Catenin Signaling-Mediated Skeletal Muscle Development by Stabilizing Dishevelled-2 Against Autophagy.

MYOF DVL2

5.49e-06282231623157
Pubmed

In Vivo and In Vitro Characterization of the RNA Binding Capacity of SETD1A (KMT2F).

SETD1A SETD1B

5.49e-06282238003223
Pubmed

Downregulation of NFAT3 Due to Lack of T-Box Transcription Factor TBX5 Is Crucial for Cytokine Expression in T Cells.

NFATC4 TBX5

5.49e-06282229180489
Pubmed

Zinc finger proteins: what we know and what we would like to know.

EGR2 GLI1

5.49e-0628221768617
Pubmed

Peroxisome proliferator-activated receptor (PPAR)-binding protein (PBP) but not PPAR-interacting protein (PRIP) is required for nuclear translocation of constitutive androstane receptor in mouse liver.

NCOA6 MED1

5.49e-06282216828057
Pubmed

A predictive model of bifunctional transcription factor signaling during embryonic tissue patterning.

GLI1 PTCH2 CDON

5.63e-061582325458012
Pubmed

The functional interactome landscape of the human histone deacetylase family.

TRERF1 NCOR2 GSE1 USP9X MDM1 SIN3A HDAC7

5.68e-0628982723752268
Pubmed

Transcription factor protein interactomes reveal genetic determinants in heart disease.

ATP5PB ZNF462 NCOR2 PIP4P1 PROSER1 SIN3A MED1 TBX5

5.91e-0641182835182466
Pubmed

Large-scale phosphomimetic screening identifies phospho-modulated motif-based protein interactions.

TRERF1 NCOR2 WASF2 SPEN RNF11

6.49e-0611082537219487
Pubmed

Proximity-dependent biotin identification (BioID) reveals a dynamic LSD1-CoREST interactome during embryonic stem cell differentiation.

TRERF1 ZNF462 PRR12 NCOR2 GSE1 ZMIZ2 DVL2 POLRMT

6.68e-0641882834709266
Pubmed

SET1 and p300 act synergistically, through coupled histone modifications, in transcriptional activation by p53.

SETD1A NCOA6 SETD1B

6.92e-061682323870121
Pubmed

H3K4 mono- and di-methyltransferase MLL4 is required for enhancer activation during cell differentiation.

SETD1A NCOA6 SETD1B

6.92e-061682324368734
Pubmed

PRISMA and BioID disclose a motifs-based interactome of the intrinsically disordered transcription factor C/EBPα.

TRERF1 PRR12 CCNT2 NCOR2 NCOA6 GSE1 BICRA PRRC2C ZMIZ2 SIN3A MED1 SPEN

1.05e-051103821234189442
Pubmed

Resetting the epigenetic balance of Polycomb and COMPASS function at enhancers for cancer therapy.

SETD1A NCOA6 SETD1B

1.40e-052082329785026
Pubmed

T0070907, a selective ligand for peroxisome proliferator-activated receptor gamma, functions as an antagonist of biochemical and cellular activities.

NCOR2 NCOA6 MED1

1.40e-052082311877444
Pubmed

FOXK2 Elicits Massive Transcription Repression and Suppresses the Hypoxic Response and Breast Cancer Carcinogenesis.

NCOR2 SETD1B SIN3A

1.40e-052082327773593
Pubmed

Nuclear receptor-coregulator interaction profiling identifies TRIP3 as a novel peroxisome proliferator-activated receptor gamma cofactor.

NCOR2 NCOA6 MED1

1.63e-052182319596656
Pubmed

WDR82, a key epigenetics-related factor, plays a crucial role in normal early embryonic development in mice.

SETD1A SETD1B

1.64e-05382221123813
Pubmed

Molecular insight into the SETD1A/B N-terminal region and its interaction with WDR82.

SETD1A SETD1B

1.64e-05382237030068
Pubmed

Smooth muscle fascicular reorientation is required for esophageal morphogenesis and dependent on Cdo.

GLI1 CDON

1.64e-05382223569214
Pubmed

Structural insights into the recruitment of SMRT by the corepressor SHARP under phosphorylative regulation.

NCOR2 SPEN

1.64e-05382224268649
Pubmed

Xp11.2 microduplications including IQSEC2, TSPYL2 and KDM5C genes in patients with neurodevelopmental disorders.

KDM5C IQSEC2

1.64e-05382226059843
Pubmed

The glucocorticoid receptor recruits the COMPASS complex to regulate inflammatory transcription at macrophage enhancers.

SETD1A SETD1B

1.64e-05382233567280
Pubmed

Structural basis for activity regulation of MLL family methyltransferases.

SETD1A NCOA6 SETD1B

1.88e-052282326886794
Pubmed

The G protein-coupled receptor Gpr161 regulates forelimb formation, limb patterning and skeletal morphogenesis in a primary cilium-dependent manner.

GLI1 SP7 TBX5

2.16e-052382329222391
Pubmed

FOXC1 and FOXC2 regulate growth plate chondrocyte maturation towards hypertrophy in the embryonic mouse limb skeleton.

GLI1 PTCH2 SP7

2.47e-052482339012257
Pubmed

Shh signaling within the dental epithelium is necessary for cell proliferation, growth and polarization.

AMBN GLI1 PTCH2

2.47e-052482312403705
Pubmed

T-box3 is a ciliary protein and regulates stability of the Gli3 transcription factor to control digit number.

GLI1 PTCH2 TBX5

2.80e-052582327046536
Pubmed

Transcriptional coactivator PRIP, the peroxisome proliferator-activated receptor gamma (PPARgamma)-interacting protein, is required for PPARgamma-mediated adipogenesis.

NCOA6 MED1

3.28e-05482212754253
Pubmed

Interaction of the Epstein-Barr virus mRNA export factor EB2 with human Spen proteins SHARP, OTT1, and a novel member of the family, OTT3, links Spen proteins with splicing regulation and mRNA export.

NCOR2 SPEN

3.28e-05482216129689
Pubmed

Wnt3a-mediated formation of phosphatidylinositol 4,5-bisphosphate regulates LRP6 phosphorylation.

DVL2 LRP6

3.28e-05482218772438
Pubmed

The pseudoreceptor BMP and activin membrane-bound inhibitor positively modulates Wnt/beta-catenin signaling.

DVL2 LRP6

3.28e-05482218838381
Pubmed

Initiation of Wnt signaling: control of Wnt coreceptor Lrp6 phosphorylation/activation via frizzled, dishevelled and axin functions.

DVL2 LRP6

3.28e-05482218077588
Pubmed

Protective neuronal induction of ATF5 in endoplasmic reticulum stress induced by status epilepticus.

ATF5 RBFOX3

3.28e-05482223518711
Pubmed

Wdpcp regulates cellular proliferation and differentiation in the developing limb via hedgehog signaling.

GLI1 SP7

3.28e-05482234225660
Pubmed

Agonist-antagonist induced coactivator and corepressor interplay on the human androgen receptor.

NCOR2 SPEN

3.28e-05482215062576
Pubmed

Role of the histone deacetylase complex in acute promyelocytic leukaemia.

NCOR2 SIN3A

3.28e-0548229486654
Pubmed

The Epigenetic Factor Landscape of Developing Neocortex Is Regulated by Transcription Factors Pax6→ Tbr2→ Tbr1.

NCOA6 SETD1B KDM5C SIN3A HDAC7

3.63e-0515782530186101
Pubmed

Loss of BAF (mSWI/SNF) chromatin-remodeling ATPase Brg1 causes multiple malformations of cortical development in mice.

RBFOX3 ROBO2 CDON

3.97e-052882335666215
Pubmed

Temporospatial sonic hedgehog signalling is essential for neural crest-dependent patterning of the intrinsic tongue musculature.

GLI1 PTCH2 CDON

3.97e-052882331719045
Pubmed

An atlas of combinatorial transcriptional regulation in mouse and man.

NCOR2 ATF5 NFATC4 GLI1 KDM5C NFKBIZ SIN3A MED1 SPEN SP7

4.10e-05877821020211142
Pubmed

Proximity-dependent Mapping of the Androgen Receptor Identifies Kruppel-like Factor 4 as a Functional Partner.

TRERF1 PRR12 NCOA6 GSE1 SIN3A MED1

4.25e-0526882633640491
Pubmed

A Retinoic Acid-Hedgehog Cascade Coordinates Mesoderm-Inducing Signals and Endoderm Competence during Lung Specification.

GLI1 PTCH2 TBX5

4.42e-052982327320915
Pubmed

The RNA-mediated estrogen receptor α interactome of hormone-dependent human breast cancer cell nuclei.

PRR12 CASC3 MYOF WASF2 ARHGEF9 POLRMT IST1 TRIOBP MED1 NDUFA8 SPEN PLEKHA7 CCDC86

4.63e-051497821331527615
Pubmed

Prediction of the coding sequences of mouse homologues of KIAA gene: II. The complete nucleotide sequences of 400 mouse KIAA-homologous cDNAs identified by screening of terminal sequences of cDNA clones randomly sampled from size-fractionated libraries.

SETD1B GSE1 PRRC2C ARHGEF9 IST1 OGFOD1 SPEN

5.10e-0540782712693553
Pubmed

Ifg, Gli, Mdm1, Mdm2, and Mdm3: candidate genes for the mouse pg locus.

GLI1 MDM1

5.47e-0558227849395
Pubmed

Biochemical reconstitution and phylogenetic comparison of human SET1 family core complexes involved in histone methylation.

SETD1A SETD1B

5.47e-05582225561738
Pubmed

Reciprocal actions of ATF5 and Shh in proliferation of cerebellar granule neuron progenitor cells.

ATF5 RBFOX3

5.47e-05582222095825
Pubmed

Components of the SMRT corepressor complex exhibit distinctive interactions with the POZ domain oncoproteins PLZF, PLZF-RARalpha, and BCL-6.

NCOR2 SIN3A

5.47e-0558229765306
Pubmed

Expression of Sonic Hedgehog and pathway components in the embryonic mouse head: anatomical relationships between regulators of positive and negative feedback.

GLI1 PTCH2

5.47e-05582234353359
Pubmed

Helicobacter pylori-induced activation of beta-catenin involves low density lipoprotein receptor-related protein 6 and Dishevelled.

DVL2 LRP6

5.47e-05582220137080
Pubmed

Mint represses transactivation of the type II collagen gene enhancer through interaction with alpha A-crystallin-binding protein 1.

NCOR2 SPEN

5.47e-05582215778499
Pubmed

RUNX1 regulates corepressor interactions of PU.1.

SIN3A CBFA2T3

5.47e-05582221518930
Pubmed

Interaction of PIMT with transcriptional coactivators CBP, p300, and PBP differential role in transcriptional regulation.

NCOA6 MED1

5.47e-05582211912212
Pubmed

Targeting fusion protein/corepressor contact restores differentiation response in leukemia cells.

NCOR2 SIN3A

5.47e-05582215729358
Pubmed

A Shh coreceptor Cdo is required for efficient cardiomyogenesis of pluripotent stem cells.

GLI1 CDON

5.47e-05582226906632
Pubmed

Expression pattern of the thrombopoietin receptor (Mpl) in the murine central nervous system.

THPO RBFOX3

5.47e-05582220667107
Pubmed

Transcription coactivator PBP, the peroxisome proliferator-activated receptor (PPAR)-binding protein, is required for PPARalpha-regulated gene expression in liver.

NCOA6 MED1

8.19e-05682215150259
Pubmed

Multipotent CD15+ cancer stem cells in patched-1-deficient mouse medulloblastoma.

GLI1 PTCH2

8.19e-05682219487286
Pubmed

CRM1 mediates nuclear export of HDAC7 independently of HDAC7 phosphorylation and association with 14-3-3s.

NCOR2 HDAC7

8.19e-05682216956611
Pubmed

Expression Profiling and Functional Analysis of Candidate Col10a1 Regulators Identified by the TRAP Program.

EGR2 TBX5

8.19e-05682234276786
Pubmed

Development gone awry: congenital heart disease.

DVL2 TBX5

8.19e-05682214976138
Pubmed

The Xist lncRNA interacts directly with SHARP to silence transcription through HDAC3.

NCOR2 SPEN

8.19e-05682225915022
Pubmed

Gli1 Regulates the Postnatal Acquisition of Peripheral Nerve Architecture.

EGR2 GLI1

8.19e-05682234772739
Pubmed

PSF is a novel corepressor that mediates its effect through Sin3A and the DNA binding domain of nuclear hormone receptors.

NCOR2 SIN3A

8.19e-05682211259580
Pubmed

Nuclear factor of activated T cells (NFAT) proteins repress canonical Wnt signaling via its interaction with Dishevelled (Dvl) protein and participate in regulating neural progenitor cell proliferation and differentiation.

NFATC4 DVL2

8.19e-05682221880741
Pubmed

Mapping Wnt/beta-catenin signaling during mouse development and in colorectal tumors.

LRP6 TBX5

8.19e-05682212626757
Pubmed

Boc modifies the spectrum of holoprosencephaly in the absence of Gas1 function.

GLI1 CDON

8.19e-05682225063195
Pubmed

Epsin is required for Dishevelled stability and Wnt signalling activation in colon cancer development.

DVL2 LRP6

8.19e-05682225871009
Pubmed

Nuclear receptor corepressors partner with class II histone deacetylases in a Sin3-independent repression pathway.

NCOR2 SIN3A

8.19e-05682210640275
Pubmed

Reciprocal interaction between SIRT6 and APC/C regulates genomic stability.

SETD1A SETD1B USP9X DVL2 TMEM209 POLRMT MED1

8.31e-0544082734244565
Pubmed

CXXC finger protein 1 contains redundant functional domains that support embryonic stem cell cytosine methylation, histone methylation, and differentiation.

SETD1A SETD1B

1.14e-04782219433449
Pubmed

Altered bone growth dynamics prefigure craniosynostosis in a zebrafish model of Saethre-Chotzen syndrome.

GLI1 SP7

1.14e-04782230375332
Pubmed

Ocular abnormalities in mice lacking the immunoglobulin superfamily member Cdo.

CDON TBX5

1.14e-04782219754878
Pubmed

A mutant with bilateral whisker to barrel inputs unveils somatosensory mapping rules in the cerebral cortex.

RBFOX3 EGR2

1.14e-04782228350297
Pubmed

The peroxisome proliferator-activated receptor delta, an integrator of transcriptional repression and nuclear receptor signaling.

NCOR2 SPEN

1.14e-04782211867749
Pubmed

Osterix is dispensable for the development of the mouse olfactory bulb.

RBFOX3 SP7

1.14e-04782227449610
InteractionEGR2 interactions

TRERF1 ZNF462 PRR12 NCOR2 NCOA6 EGR2 BICRA ZMIZ2 PROSER1

3.18e-08171829int:EGR2
InteractionRUNX1T1 interactions

NCOR2 GSE1 DVL2 SIN3A PLSCR3 CBFA2T3 SPEN TBX5

4.80e-08127828int:RUNX1T1
InteractionKDM6A interactions

SETD1A NCOA6 SETD1B EGR2 KDM5C PROSER1 SP7 TBX5

3.15e-07162828int:KDM6A
InteractionSP7 interactions

TRERF1 PRR12 NCOR2 NCOA6 GSE1 BICRA ZMIZ2 PROSER1 SIN3A SP7

4.32e-073048210int:SP7
InteractionEYA4 interactions

PRR12 NCOR2 GSE1 BICRA ZMIZ2 CCDC120 PROSER1 VPS37B SP7

6.33e-07243829int:EYA4
InteractionHNF4A interactions

ZNF462 PRR12 SETD1A NCOR2 NCOA6 GSE1 BICRA MED1 SPEN

1.77e-06275829int:HNF4A
InteractionNCOA6 interactions

SETD1A NCOR2 NCOA6 SETD1B EGR2 MED1 SP7

2.09e-06145827int:NCOA6
InteractionTLE3 interactions

TRERF1 PRR12 NCOR2 CRTC3 GSE1 EGR2 ZMIZ2 PROSER1 SPEN SP7

2.94e-063768210int:TLE3
InteractionKDM1A interactions

TRERF1 ATP5PB ZNF462 PRR12 NCOR2 GSE1 USP9X DVL2 POLRMT SIN3A NDUFA8 CBFA2T3 VPS37B SP7 TBX5

5.19e-069418215int:KDM1A
InteractionNUP35 interactions

PRR12 NCOR2 NCOA6 CRTC3 GSE1 PRRC2C GLI1 TMEM209 POLRMT TBX5

8.47e-064248210int:NUP35
InteractionCRX interactions

TRERF1 ZNF462 PRR12 NCOR2 BICRA ZMIZ2 PROSER1 SPEN

9.09e-06254828int:CRX
InteractionGUSBP5 interactions

NCOR2 GSE1 KDM5C DVL2 SPEN

1.36e-0575825int:GUSBP5
InteractionPAX9 interactions

PRR12 NCOR2 NCOA6 GSE1 ZMIZ2 PROSER1

1.50e-05130826int:PAX9
InteractionNCOR1 interactions

NCOR2 EGR2 KDM5C SIN3A CBFA2T3 SPEN HDAC7 TRIM52 SP7

1.66e-05363829int:NCOR1
InteractionFEV interactions

ZNF462 PRR12 SETD1A NCOR2 NCOA6 GSE1 BICRA

1.90e-05203827int:FEV
InteractionYAP1 interactions

TRERF1 WBP1 SETD1A NCOA6 CRTC3 PRRC2C GLI1 USP9X PIP4P1 TRIOBP CCDC120 SIN3A MED1 SPEN RNF11

3.12e-0510958215int:YAP1
InteractionRERE interactions

SETD1A SETD1B EGR2 CCDC120 SP7

3.87e-0593825int:RERE
InteractionNFIX interactions

PRR12 SETD1A NCOR2 GSE1 BICRA SPEN SP7

3.89e-05227827int:NFIX
InteractionSHH interactions

PTCH2 SIN3A CDON

5.07e-0518823int:SHH
InteractionSOX5 interactions

NCOR2 GSE1 EGR2 PRRC2C PROSER1 SP7

5.20e-05162826int:SOX5
InteractionIRF2BP2 interactions

NCOR2 SIN3A CBFA2T3 SPEN SP7

8.64e-05110825int:IRF2BP2
InteractionZMYND10 interactions

NUTM1 WBP1 TBX5

9.46e-0522823int:ZMYND10
InteractionTBR1 interactions

PRR12 NCOR2 GSE1 PROSER1 SP7

9.81e-05113825int:TBR1
InteractionITCH interactions

TRERF1 WBP1 GLI1 USP9X DVL2 LRP6 SPEN RNF11

1.00e-04356828int:ITCH
InteractionNCOR2 interactions

NCOR2 NCOA6 EGR2 SIN3A SPEN HDAC7 SP7

1.01e-04264827int:NCOR2
InteractionTBXT interactions

PRR12 NCOR2 NCOA6 GSE1 SPEN

1.11e-04116825int:TBXT
InteractionFLI1 interactions

EGR2 USP9X SOX30 SP7

1.19e-0462824int:FLI1
InteractionHNF1B interactions

PRR12 NCOR2 GSE1 BICRA PROSER1 SP7

1.25e-04190826int:HNF1B
InteractionEP300 interactions

TRERF1 NUTM1 CASC3 SETD1A NCOR2 NCOA6 ZNF469 ATF5 THPO EGR2 USP9X DVL2 SIN3A MED1 HDAC7 SP7

1.43e-0414018216int:EP300
InteractionRBBP5 interactions

CCNT2 SETD1A NCOA6 SETD1B EGR2 SIN3A SPEN

1.69e-04287827int:RBBP5
InteractionNR1H2 interactions

NCOR2 NCOA6 ROBO2 MED1

1.70e-0468824int:NR1H2
InteractionTLX3 interactions

PRR12 NCOR2 NCOA6 GSE1 ZMIZ2 PROSER1 TOX2

1.84e-04291827int:TLX3
InteractionHCFC1 interactions

SETD1A NCOA6 SETD1B EGR2 PRRC2C SIN3A TBX5

1.92e-04293827int:HCFC1
InteractionHDAC4 interactions

PRR12 NCOR2 SETD1B RBFOX3 EGR2 PRRC2C USP9X WASF2 SIN3A PLEKHA7 HDAC7

2.07e-047448211int:HDAC4
InteractionKMT2C interactions

SETD1A NCOA6 SETD1B EGR2 SP7

2.18e-04134825int:KMT2C
InteractionNUP43 interactions

ZNF462 CCNT2 SETD1A NCOR2 NCOA6 SETD1B GSE1 PRRC2C KDM5C SPEN

2.20e-046258210int:NUP43
InteractionGATA4 interactions

ATP5PB ZNF462 NCOR2 NFATC4 PIP4P1 PROSER1 MED1 TBX5

2.67e-04411828int:GATA4
InteractionPROSER1 interactions

EGR2 PROSER1 SP7

2.69e-0431823int:PROSER1
InteractionFOXQ1 interactions

ATP5PB NCOR2 GSE1 POLRMT CCDC86

2.76e-04141825int:FOXQ1
InteractionERG interactions

PRR12 NCOR2 NCOA6 GSE1 BICRA USP9X

2.98e-04223826int:ERG
InteractionTRERF1 interactions

TRERF1 EGR2 SP7

3.24e-0433823int:TRERF1
InteractionTRB interactions

NCOA6 DVL2

3.39e-047822int:TRB
InteractionBCL6 interactions

ATP5PB NCOR2 ARHGEF9 DVL2 SIN3A HDAC7

3.44e-04229826int:BCL6
InteractionDTX2 interactions

PRR12 NCOR2 CRTC3 GSE1 TMEM209 CCDC120 PLEKHA7

3.94e-04330827int:DTX2
InteractionPBX1 interactions

USP9X CCDC120 SP7 TBX5

4.01e-0485824int:PBX1
InteractionSOX6 interactions

NCOR2 GSE1 PRRC2C ZMIZ2 PROSER1

4.53e-04157825int:SOX6
InteractionCEBPA interactions

TRERF1 PRR12 CCNT2 NCOR2 NCOA6 ATF5 GSE1 NFATC4 BICRA PRRC2C ZMIZ2 SIN3A MED1 SPEN

4.63e-0412458214int:CEBPA
InteractionHDAC1 interactions

TRERF1 NCOR2 GSE1 FOLH1 GLI1 KDM5C ZMIZ2 DVL2 POLRMT SIN3A CBFA2T3 SPEN HDAC7

5.07e-0411088213int:HDAC1
InteractionTRIM33 interactions

EGR2 USP9X KDM5C DVL2 CBFA2T3 TRIM52 SP7 TBX5

5.10e-04453828int:TRIM33
InteractionPRMT2 interactions

SETD1A NCOA6 SETD1B IQSEC2

5.20e-0491824int:PRMT2
InteractionNFKBIL1 interactions

SETD1A USP9X DVL2 SPEN

5.65e-0493824int:NFKBIL1
InteractionZNF608 interactions

SETD1A SETD1B EGR2 SP7

5.65e-0493824int:ZNF608
GeneFamilyX-linked mental retardation|Angiotensin receptors

USP9X KDM5C IQSEC2

5.91e-0453563103
CoexpressionGSE28737_WT_VS_BCL6_HET_MARGINAL_ZONE_BCELL_UP

DDR1 SETD1B GSE1 ERN1 DTNB GLI1 PIP4P1

3.18e-06200827M9342
CoexpressionGSE9946_LISTERIA_INF_MATURE_VS_PROSTAGLANDINE2_TREATED_MATURE_DC_UP

SETD1A NCOR2 MDM1 SIN3A SPEN TRIM52

4.06e-06134826M430
CoexpressionGSE37532_VISCERAL_ADIPOSE_TISSUE_VS_LN_DERIVED_TREG_CD4_TCELL_DN

SETD1A CRTC3 BICRA WASF2 OGFOD1 PLEKHA7

9.38e-06155826M8944
CoexpressionGSE23925_LIGHT_ZONE_VS_NAIVE_BCELL_UP

PTPRN EGR2 CASKIN2 IST1 NFKBIZ VPS37B

3.85e-05199826M7885
CoexpressionGSE12198_CTRL_VS_HIGH_IL2_STIM_NK_CELL_DN

EGR2 NFATC4 CASKIN2 GLI1 CCDC86 HDAC7

3.96e-05200826M7070
CoexpressionGSE28237_FOLLICULAR_VS_EARLY_GC_BCELL_UP

CCNT2 NCOR2 PTPRN LRP6 MED1 CBFA2T3

3.96e-05200826M4884
DrugSulconazole nitrate [61318-91-0]; Up 200; 8.6uM; MCF7; HT_HG-U133A

NCOR2 MYOF NFATC4 DTNB PTCH2 TJAP1 TBX5

5.03e-061898173373_UP
Drugwortmannin from Penicillium funiculosum; Down 200; 0.01uM; HL60; HT_HG-U133A

MYOF ATF5 THPO ARHGEF9 DVL2 LRP6 PLSCR3

5.58e-061928172703_DN
DrugNaltrexone hydrochloride dihydrate [16676-29-2]; Down 200; 9.6uM; MCF7; HT_HG-U133A

GPR137 SETD1A AMPD3 IQSEC2 LRP6 TJAP1 SPEN

5.77e-061938172209_DN
DrugTridihexethyl chloride; Up 200; 11.4uM; MCF7; HT_HG-U133A

GPR137 SETD1A BICRA ZMIZ2 HDAC7 CDON TBX5

5.97e-061948173526_UP
DrugGSK-3 Inhibitor IX; Up 200; 0.5uM; PC3; HT_HG-U133A

SETD1A ATF5 NFATC4 CASKIN2 PRRC2C ZMIZ2 TRIOBP

6.39e-061968176559_UP
DrugCefotaxime sodium salt [64485-93-4]; Down 200; 8.4uM; PC3; HT_HG-U133A

GPR137 MYOF AMPD3 CASKIN2 KDM5C MDM1 ARHGEF9

6.61e-061978172072_DN
DrugMethyldopate hydrochloride [2508-79-4]; Up 200; 14.6uM; MCF7; HT_HG-U133A

GPR137 AMPD3 CASKIN2 ZMIZ2 IQSEC2 LRP6 HDAC7

7.06e-061998174986_UP
Drugrosiglitazone; Down 200; 10uM; HL60; HT_HG-U133A

NCOR2 MYOF IQSEC2 KHDRBS2 ARHGEF9 DVL2 CDON

7.06e-061998172693_DN
DrugLY 294002; Down 200; 0.1uM; HL60; HT_HG-U133A

SETD1A NCOR2 MYOF THPO KHDRBS2 LRP6 CDON

7.06e-061998172676_DN
Drug4-(4-(2,3-dihydrobenzo(1,4)dioxin-6-yl)-5-pyridin-2-yl-1H-imidazol-2-yl)benzamide

DVL2 LRP6

3.74e-053812ctd:C493177
Drugscriptaid; Down 200; 10uM; PC3; HT_HG-U133A

CCNT2 MYOF ARHGEF9 TRIOBP MED1 HDAC7

4.74e-051828166896_DN
DrugMexiletine hydrochloride [5370-01-4]; Down 200; 18.6uM; PC3; HT_HG-U133A

GPR137 SETD1A CASKIN2 ZMIZ2 TMEM209 TJAP1

6.57e-051938164338_DN
DrugPimethixene maleate [13187-06-9]; Down 200; 9.8uM; MCF7; HT_HG-U133A

SETD1A MDM1 ARHGEF9 LRP6 PLSCR3 MED1

6.76e-051948167468_DN
DrugFludrocortisone acetate [514-36-3]; Down 200; 9.4uM; MCF7; HT_HG-U133A

AMPD3 KDM5C ZMIZ2 SOX30 DVL2 TBX5

6.76e-051948163977_DN
DrugCP-690334-01 [459212-38-5]; Up 200; 10uM; MCF7; HT_HG-U133A

GPR137 SETD1B DTNB SOX30 TJAP1 CDON

6.76e-051948163906_UP
Drug2-Chloropyrazine [14508-49-7]; Down 200; 35uM; MCF7; HT_HG-U133A

CCNT2 AMPD3 CASKIN2 KDM5C ARHGEF9 TRIOBP

6.76e-051948163570_DN
DrugClozapine [5786-21-0]; Up 200; 12.2uM; MCF7; HT_HG-U133A

GPR137 SETD1A NCOR2 DVL2 HDAC7 TBX5

6.96e-051958165265_UP
DrugCinchonine [118-10-5]; Up 200; 13.6uM; MCF7; HT_HG-U133A

GPR137 NFATC4 ZMIZ2 TMEM209 CDON TBX5

6.96e-051958164107_UP
DrugFenoprofen calcium salt dihydrate [53746-45-5]; Down 200; 7.2uM; PC3; HT_HG-U133A

GPR137 NCOR2 SETD1B ZMIZ2 IQSEC2 DVL2

6.96e-051958163714_DN
DrugEthamsylate [2624-44-4]; Down 200; 15.2uM; MCF7; HT_HG-U133A

GPR137 CCNT2 ZMIZ2 IQSEC2 TJAP1 HDAC7

6.96e-051958164399_DN
DrugOxamniquine [21738-42-1]; Up 200; 14.4uM; MCF7; HT_HG-U133A

NCOR2 AMPD3 KHDRBS2 PLSCR3 CDON TBX5

6.96e-051958164124_UP
DrugFinasteride [98319-26-7]; Up 200; 10.8uM; MCF7; HT_HG-U133A

GPR137 AMPD3 NFATC4 SOX30 TMEM209 TJAP1

7.16e-051968166062_UP
DrugSulpiride [15676-16-1]; Down 200; 11.8uM; MCF7; HT_HG-U133A

CCNT2 MYOF ZMIZ2 DVL2 TJAP1 HDAC7

7.16e-051968164389_DN
DrugOrphenadrine hydrochloride [341-69-5]; Down 200; 13uM; MCF7; HT_HG-U133A

SETD1A MYOF AMPD3 TMEM209 TJAP1 PLSCR3

7.16e-051968162318_DN
DrugHydroflumethiazide [135-09-1]; Up 200; 12uM; MCF7; HT_HG-U133A

GPR137 MYOF IQSEC2 TJAP1 PLSCR3 CDON

7.16e-051968161687_UP
DrugTetracaone hydrochloride [136-47-0]; Up 200; 13.2uM; MCF7; HT_HG-U133A

GPR137 MYOF DTNB ZMIZ2 IQSEC2 PLSCR3

7.36e-051978162888_UP
DrugQuinic acid [86-68-0]; Up 200; 19.6uM; MCF7; HT_HG-U133A

GPR137 SETD1A ERN1 NFATC4 TMEM209 PLSCR3

7.36e-051978163540_UP
DrugBenzamil hydrochloride [2898-76-2]; Up 200; 11.2uM; MCF7; HT_HG-U133A

GPR137 AMPD3 SETD1B ERN1 NFATC4 TBX5

7.36e-051978164760_UP
DrugSpaglumic acid [4910-46-7]; Down 200; 13.2uM; MCF7; HT_HG-U133A

SETD1A CASKIN2 ARHGEF9 DVL2 TMEM209 PLSCR3

7.36e-051978167465_DN
DrugNS-398; Down 200; 10uM; MCF7; HT_HG-U133A

KDM5C ZMIZ2 IQSEC2 DVL2 TRIOBP PLSCR3

7.36e-051978166897_DN
Drugestradiol, USP; Up 200; 0.1uM; PC3; HT_HG-U133A

GPR137 CCNT2 ZMIZ2 ARHGEF9 TMEM209 TJAP1

7.57e-051988161208_UP
DrugNafcillin sodium salt monohydrate [7177-50-6]; Down 200; 8.8uM; HL60; HT_HG-U133A

GPR137 THPO ZMIZ2 KHDRBS2 LRP6 HDAC7

7.57e-051988162983_DN
Drug0173570-0000 [211245-44-2]; Up 200; 1uM; PC3; HT_HG-U133A

GPR137 CCNT2 NCOR2 ZMIZ2 ARHGEF9 TJAP1

7.57e-051988167391_UP
DrugFamotidine [76824-35-6]; Up 200; 11.8uM; MCF7; HT_HG-U133A

GPR137 CCNT2 ERN1 MED1 CDON TBX5

7.57e-051988161529_UP
DrugHeptaminol hydrochloride [543-15-7]; Down 200; 22uM; PC3; HT_HG-U133A

MYOF ZMIZ2 ARHGEF9 MED1 SPEN HDAC7

7.57e-051988161825_DN
Drugnordihydroguaiaretic acid; Down 200; 1uM; HL60; HT_HG-U133A

GPR137 SETD1A NCOR2 MYOF KHDRBS2 TJAP1

7.78e-051998162683_DN
DrugCarbamazepine [298-46-4]; Up 200; 17uM; HL60; HT_HG-U133A

GPR137 MYOF KDM5C PLSCR3 HDAC7 CDON

7.78e-051998161847_UP
DrugPalmatine chloride [3486-67-7]; Up 200; 10.4uM; MCF7; HT_HG-U133A

CCNT2 NCOR2 ERN1 DTNB LRP6 HDAC7

7.78e-051998164957_UP
DrugCarbenoxolone disodium salt [7421-40-1]; Down 200; 6.6uM; HL60; HT_HG-U133A

THPO ZMIZ2 IQSEC2 TMEM209 PLSCR3 HDAC7

8.00e-052008163014_DN
DrugMidodrine hydrochloride [3092-17-9]; Up 200; 13.8uM; PC3; HT_HG-U133A

GPR137 ATF5 BICRA KHDRBS2 DVL2 MED1

8.00e-052008167156_UP
DrugMethamphetamine

NCOR2 AMPD3 THPO ERN1 EGR2 NFATC4 PRRC2C GLI1 WASF2 ZMIZ2 OBSCN IST1 TJAP1 VPS37B HDAC7

1.11e-0414018115ctd:D008694
DrugR)-3-pyrrolidinecarboxylic acid

THPO DTNB

1.86e-046812CID001501969
Drugvinylene

ZNF462 NCOR2 EGR2 GLI1 ARHGEF9 SP7

2.42e-04245816CID000006326
Drugguvacoline

NUTM1 THPO

2.59e-047812CID000160492
DrugTrichostatin A, from Streptomyces sp.; Down 200; 0.1uM; MCF7; HT_HG-U133A

MYOF ATF5 SETD1B CASKIN2 CBFA2T3

3.27e-041678153979_DN
DrugTrichostatin A, from Streptomyces sp.; Down 200; 0.1uM; PC3; HT_HG-U133A

SETD1B CASKIN2 ARHGEF9 TRIOBP HDAC7

3.94e-041748153993_DN
DrugTrichostatin A, Streptomyces sp.; Down 200; 1uM; MCF7; HT_HG-U133A

NCOA6 ATF5 SETD1B GSE1 CBFA2T3

3.94e-041748151659_DN
Drugtrichostatin A, Streptomyces sp.; Down 200; 1uM; MCF7; HT_HG-U133A

GPR137 NCOR2 MYOF SETD1B CBFA2T3

4.16e-041768155976_DN
Drugtrichostatin A, Streptomyces sp.; Down 200; 1uM; PC3; HT_HG-U133A

MYOF ATF5 SETD1B MED1 HDAC7

4.27e-041778157047_DN
DrugGANT 61

GLI1 KHDRBS2

4.43e-049812ctd:C551027
Drug2-methoxy-5-nitrotropone

ELL2 DTNB

4.43e-049812CID000084563
DrugNSC53670

EGR2 GLI1 KHDRBS2

5.17e-0444813CID000243583
DrugRapamycin; Up 200; 0.1uM; MCF7; HT_HG-U133A_EA

MYOF ARHGEF9 DVL2 TJAP1 HDAC7

5.22e-041858151022_UP
DrugFlumethasone [2135-17-3]; Up 200; 9.8uM; HL60; HT_HG-U133A

NCOR2 DTNB ARHGEF9 PTCH2 PLSCR3

5.22e-041858152551_UP
DrugLithocholic acid [434-13-9]; Up 200; 10.6uM; HL60; HT_HG-U133A

MYOF ERN1 ARHGEF9 LRP6 TJAP1

5.48e-041878152571_UP
Drugtroglitazone; Down 200; 10uM; HL60; HT_HG-U133A

NCOR2 MYOF ZMIZ2 ARHGEF9 TJAP1

5.75e-041898152692_DN
DrugEthisterone [434-03-7]; Down 200; 12.8uM; PC3; HT_HG-U133A

GPR137 CCNT2 NCOR2 KDM5C ZMIZ2

5.89e-041908154340_DN
DrugFluvoxamine maleate [61718-82-9]; Down 200; 9.2uM; MCF7; HT_HG-U133A

GPR137 AMPD3 PRRC2C TMEM209 LRP6

5.89e-041908154114_DN
Drug0317956-0000 [391210-11-0]; Down 200; 1uM; PC3; HT_HG-U133A

GPR137 NCOR2 CASKIN2 ZMIZ2 TJAP1

6.17e-041928154334_DN
DrugCyanocobalamin [68-19-9]; Down 200; 3uM; MCF7; HT_HG-U133A

PRRC2C TMEM209 LRP6 TJAP1 PLSCR3

6.17e-041928153252_DN
DrugPHA-00851261E [724719-49-7]; Down 200; 10uM; PC3; HT_HG-U133A

GPR137 SETD1A CASKIN2 DVL2 HDAC7

6.17e-041928154330_DN
DrugNefopam hydrochloride [23327-57-3]; Down 200; 13.8uM; MCF7; HT_HG-U133A

GPR137 IQSEC2 DVL2 PLSCR3 HDAC7

6.32e-041938153627_DN
DrugLevodopa [59-92-7]; Down 200; 20.2uM; MCF7; HT_HG-U133A

GPR137 CCNT2 ZMIZ2 TJAP1 HDAC7

6.32e-041938154394_DN
DrugProbenecid [57-66-9]; Down 200; 14uM; MCF7; HT_HG-U133A

AMPD3 ATF5 CASKIN2 BICRA TMEM209

6.32e-041938152825_DN
DrugHymecromone [90-33-5]; Down 200; 22.8uM; PC3; HT_HG-U133A

NCOR2 DTNB KDM5C IQSEC2 TJAP1

6.32e-041938154623_DN
Drug5114445; Down 200; 10uM; MCF7; HT_HG-U133A_EA

ATF5 CASKIN2 PRRC2C TRIOBP SPEN

6.32e-04193815901_DN
DrugProgesterone [57-83-0]; Down 200; 12.8uM; PC3; HT_HG-U133A

MYOF CASKIN2 BICRA TJAP1 HDAC7

6.32e-041938156646_DN
DrugHydrochlorothiazide [58-93-5]; Down 200; 13.4uM; PC3; HT_HG-U133A

MDM1 LRP6 TJAP1 PLSCR3 CDON

6.32e-041938156625_DN
DrugAmiodarone hydrochloride [19774-82-4]; Up 200; 5.8uM; MCF7; HT_HG-U133A

CCNT2 MYOF AMPD3 CDON TBX5

6.32e-041938153296_UP
DrugLY 294002; Down 200; 10uM; MCF7; HT_HG-U133A

GPR137 ATF5 CASKIN2 TMEM209 CCDC86

6.47e-041948155587_DN
DrugNystatine [1400-61-9]; Up 200; 4.4uM; PC3; HT_HG-U133A

GPR137 AMPD3 CASKIN2 ZMIZ2 IQSEC2

6.47e-041948154223_UP
DrugBetahistine mesylate [54856-23-4]; Down 200; 17.2uM; HL60; HT_HG-U133A

CCNT2 MYOF ARHGEF9 TMEM209 TJAP1

6.47e-041948152472_DN
Drug0317956-0000 [391210-11-0]; Down 200; 10uM; PC3; HT_HG-U133A

GPR137 CASKIN2 KDM5C ZMIZ2 HDAC7

6.47e-041948154331_DN
DrugFlutamide [13311-84-7]; Down 200; 14.4uM; MCF7; HT_HG-U133A

PRRC2C ZMIZ2 TMEM209 LRP6 MED1

6.47e-041948154361_DN
DrugGallamine triethiodide [65-29-2]; Down 200; 4.4uM; MCF7; HT_HG-U133A

GPR137 MYOF CASKIN2 LRP6 CDON

6.47e-041948152221_DN
DrugEtifenin [63245-28-3]; Up 200; 12.4uM; MCF7; HT_HG-U133A

MYOF CASKIN2 TMEM209 PLSCR3 TBX5

6.47e-041948154117_UP
DrugTolbutamide [64-77-7]; Up 200; 14.8uM; PC3; HT_HG-U133A

THPO ERN1 DTNB KHDRBS2 TJAP1

6.62e-041958153804_UP
DrugSisomicin sulfate [53179-09-2]; Up 200; 2.8uM; MCF7; HT_HG-U133A

DTNB ZMIZ2 DVL2 HDAC7 TBX5

6.62e-041958152853_UP
DrugBumetanide [28395-03-1]; Down 200; 11uM; HL60; HT_HG-U133A

DVL2 TMEM209 LRP6 PLSCR3 MED1

6.62e-041958152409_DN
DrugKawain [500-64-1]; Down 200; 17.4uM; PC3; HT_HG-U133A

GPR137 SETD1A NCOR2 ZMIZ2 CDON

6.62e-041958153670_DN
DrugDrofenine hydrochloride [548-66-3]; Up 200; 11.4uM; MCF7; HT_HG-U133A

GPR137 CCNT2 IQSEC2 KHDRBS2 MED1

6.62e-041958153455_UP
DrugClomiphene citrate (Z,E) [50-41-9]; Up 200; 6.6uM; MCF7; HT_HG-U133A

PTPRN ZMIZ2 IQSEC2 DVL2 HDAC7

6.62e-041958152624_UP
DrugOfloxacin [82419-36-1]; Up 200; 11uM; PC3; HT_HG-U133A

GPR137 NCOR2 CASKIN2 IQSEC2 TJAP1

6.62e-041958157372_UP
DrugCephalexin monohydrate [23325-78-2]; Up 200; 11uM; HL60; HT_HG-U133A

CCNT2 ATF5 ZMIZ2 PLSCR3 HDAC7

6.62e-041958151273_UP
DrugEstradiol-17 beta [50-28-2]; Up 200; 14.6uM; MCF7; HT_HG-U133A

MYOF AMPD3 IQSEC2 LRP6 PLSCR3

6.62e-041958152653_UP
DrugAmprolium hydrochloride [137-88-2]; Up 200; 12.6uM; MCF7; HT_HG-U133A

NCOR2 ZMIZ2 IQSEC2 TMEM209 TJAP1

6.78e-041968151479_UP
DrugCephapirin sodium salt [24356-60-3]; Down 200; 9uM; PC3; HT_HG-U133A

GPR137 MYOF ARHGEF9 TMEM209 LRP6

6.78e-041968157142_DN
DrugMetanephrine hydrochloride DL [881-95-8]; Up 200; 17.2uM; MCF7; HT_HG-U133A

GPR137 AMPD3 TMEM209 TJAP1 TBX5

6.78e-041968151515_UP
DrugPrilocaine hydrochloride [1786-81-8]; Down 200; 15.6uM; MCF7; HT_HG-U133A

MYOF AMPD3 ZMIZ2 IQSEC2 DVL2

6.78e-041968152314_DN
DrugQuinic acid [86-68-0]; Down 200; 19.6uM; PC3; HT_HG-U133A

NCOR2 MYOF BICRA DVL2 CDON

6.78e-041968157317_DN
DrugNialamide [51-12-7]; Down 200; 13.4uM; MCF7; HT_HG-U133A

AMPD3 SETD1B KDM5C ZMIZ2 PLSCR3

6.78e-041968154347_DN
DrugIoxaglic acid [59017-64-0]; Down 200; 3.2uM; MCF7; HT_HG-U133A

CCNT2 SETD1B DVL2 TMEM209 LRP6

6.78e-041968157470_DN
DrugAmphotericin B [1397-89-3]; Down 200; 4.4uM; MCF7; HT_HG-U133A

CASKIN2 TMEM209 TRIOBP LRP6 PLSCR3

6.78e-041968155404_DN
DrugPNU-0230031 [267429-39-0]; Up 200; 10uM; PC3; HT_HG-U133A

NFATC4 ZMIZ2 IQSEC2 DVL2 TJAP1

6.78e-041968153732_UP
DrugTrifluoperazine dihydrochloride [440-17-5]; Up 200; 8.4uM; HL60; HT_HG-U133A

ZMIZ2 IQSEC2 ARHGEF9 PLSCR3 HDAC7

6.78e-041968152389_UP
DrugMeglumine [6284-40-8]; Down 200; 20.4uM; MCF7; HT_HG-U133A

GPR137 AMPD3 ZMIZ2 KHDRBS2 LRP6

6.78e-041968156445_DN
DrugOfloxacin [82419-36-1]; Down 200; 11uM; PC3; HT_HG-U133A

SETD1A NCOR2 CASKIN2 ZMIZ2 CDON

6.78e-041968153673_DN
DrugTracazolate hydrochloride [41094-88-6]; Down 200; 11.8uM; PC3; HT_HG-U133A

GPR137 ZMIZ2 LRP6 HDAC7 CDON

6.78e-041968156619_DN
DrugFenofibrate [49562-28-9]; Up 200; 11uM; MCF7; HT_HG-U133A

GPR137 CCNT2 ZMIZ2 MED1 TRIM52

6.78e-041968157432_UP
DrugTimolol maleate salt [26921-17-5]; Down 200; 9.2uM; MCF7; HT_HG-U133A

MYOF CASKIN2 ZMIZ2 IQSEC2 KHDRBS2

6.78e-041968156483_DN
Diseaseneurodevelopmental disorder with speech impairment and dysmorphic facies (implicated_via_orthology)

SETD1A SETD1B

7.08e-062792DOID:0070417 (implicated_via_orthology)
DiseaseEpilepsy

SETD1A ERN1 KDM5C IQSEC2

2.14e-04109794C0014544
DiseaseGastrointestinal Stromal Sarcoma

GLI1 PTCH2 CDON

2.75e-0447793C3179349
Diseaseglucagon-like peptide-1 measurement

AMBN BICRA

3.14e-0410792EFO_0008465
DiseaseGastrointestinal Stromal Tumors

GLI1 PTCH2 CDON

3.31e-0450793C0238198
DiseaseDiffuse Large B-Cell Lymphoma

GLI1 SPEN CCDC86

4.38e-0455793C0079744
Diseasetestosterone measurement

CASC3 NCOR2 DDR1 NCOA6 AMPD3 EGR2 IQSEC2 CNKSR3 ARHGEF9 SIN3A PLSCR3

5.73e-0412757911EFO_0004908
Diseasevision disorder

THPO RBFOX3

8.29e-0416792MONDO_0021084
Diseasecolorectal cancer (is_marker_for)

DDR1 GLI1 KDM5C HDAC7

8.50e-04157794DOID:9256 (is_marker_for)
DiseasePR interval

ZNF469 CASKIN2 CNKSR3 OBSCN TJAP1 TBX5

2.14e-03495796EFO_0004462
Diseaseintraocular pressure measurement

MYOF ZNF469 FOLH1 PTCH2 TRIOBP PLEKHA7

2.46e-03509796EFO_0004695
DiseaseHodgkins lymphoma, multiple myeloma, chronic lymphocytic leukemia

ELL2 DTNB

2.56e-0328792EFO_0000095, EFO_0000183, EFO_0001378

Protein segments in the cluster

PeptideGeneStartEntry
VFNHPLPPPPPVTYQ

CCNT2

661

O60583
PPLPSTYLPISHPPQ

ELL2

376

O00472
QHQLPPVPGSPEPYP

CCDC86

151

Q9H6F5
YSLPVHPPPLPSQPS

AMBN

101

Q9NP70
PLLPPPPQNSVPHYA

DDR1

556

Q08345
YPIPTPGSLPPLHPS

GSE1

281

Q14687
PAPHPYSPQPPPYHE

DVL2

556

O14641
TGQPHLVPVPPLPEY

ATP5PB

36

P24539
ARSVPPSYPPPQDPL

ARHGEF9

461

O43307
PDFHPPPLPQEDPYC

AMPD3

196

Q01432
PPQPSRLAPYPHPAT

ATF5

191

Q9Y2D1
NGIPAEYAPPPPHPT

RBFOX3

16

A6NFN3
LDHLYSPPPPPPPYS

EGR2

161

P11161
PNYFEPPIPRSPHIP

OGFOD1

246

Q8N543
PPSDLYLPPPDHGAP

NCOR2

2176

Q9Y618
PPQPPHPSLSYEPAL

PTPRN

191

Q16849
SPFPIPPQSPAYEPN

NFKBIZ

311

Q9BYH8
TPPHRRDPPPSPTEY

GPR137

356

Q96N19
SPLPLYSPAPQHPPA

IQSEC2

1366

Q5JU85
PPPPGYENVSDIVPP

FOLH1

146

Q04609
PPTARAYPPPHPNQA

CCDC120

86

Q96HB5
PPYPVTPGYPEPALH

PLSCR3

16

Q9NRY6
YPTNPPGQLPSPPHV

MDM1

621

Q8TC05
NYDSEPVPPPPTPRS

LRP6

1561

O75581
PPHPQPLFSHYPQPS

GLI1

841

P08151
ALPPPPPPHQVSYDY

FAM181B

381

A6NEQ2
NGPPQPTPPPHYRLE

CBFA2T3

331

O75081
PQPPAEEPPHPLTYS

CASKIN2

371

Q8WXE0
PALPFLPPTSDPPDH

NUTM1

26

Q86Y26
STYNPHKPVPYPIPP

PROSER1

191

Q86XN7
DPSQPPPPPLQHYLE

OBSCN

5816

Q5VST9
VQTPSHPPPPYPFGS

NCOA6

366

Q14686
LDLEEFVPPVPPPPY

FAM189B

236

P81408
ALPPPPPPHLYPNTQ

CASC3

641

O15234
YFHEPPEPQPPVTPD

ERN1

961

O75460
QVSPPPPYPAPQELT

CRTC3

441

Q6UUV7
SPPPVVPVVAPYPQD

CDON

1131

Q4KMG0
PTREPPHPVFPEQPE

DTNB

311

O60941
PNIHPPQIPATPPSY

IST1

266

P53990
PTVPGYRAPPPPAHE

KHDRBS2

251

Q5VWX1
PVPSLPSDPPEHFPL

HDAC7

136

Q8WUI4
TPASPPPLHRPEAYP

BICRA

1531

Q9NZM4
PPGPQSPEHPPTTIY

C4orf54

1546

D6RIA3
VPAPPSEAPQPPEAH

POLRMT

731

O00411
PLPENPYHSRPRPDP

NDUFA8

136

P51970
HPAVLPGEDPPPYSP

PIP4P1

56

Q86T03
STPPTTYPQPVPHPQ

MED1

746

Q15648
PPPPYQEQVPVPVYH

RNF11

36

Q9Y3C5
PPPEDAPLYPHSPGS

USP9X

2491

Q93008
PPPQPPTPDYTESDI

SHD

16

Q96IW2
PPPNPYPLPQEHSQI

TBX5

306

Q99593
SPPRPPYPSYPHEDP

NFATC4

716

Q14934
PPPLPGAYIHPAPDE

PTCH2

1166

Q9Y6C5
IPEPPPVSFQPYHPL

TENT5D

366

Q8NEK8
PELYSPEDQPPAVPP

PLEKHA7

926

Q6IQ23
SSTVPPPPHRPLYQP

PRRC2C

706

Q9Y520
PYASPRSPPVQPHTP

SIN3A

271

Q96ST3
QTPVAHFPPPPEEPT

SETD1B

401

Q9UPS6
HYQRPASAQPPPPPP

PRR12

291

Q9ULL5
DFLPVVPHPYEPPEP

PROB1

686

E7EW31
PPHQPAYLLPPRPDG

SETD1A

626

O15047
APESEPPHHEPPYIP

TRIOBP

1046

Q9H2D6
PPHHEPPYIPPAVCI

TRIOBP

1051

Q9H2D6
PQASPIPHPHVYQPP

SOX30

581

O94993
IPPPPAVPYSPRDEN

CNK3/IPCEF1

346

G9CGD6
IPPPPAVPYSPRDEN

CNKSR3

346

Q6P9H4
EKLNPYPTPSPPHPL

TJAP1

311

Q5JTD0
YPDIHPPPSLPLPGQ

TRIM52

166

Q96A61
YEPSTPEPPPQVPAL

RBP3

91

P10745
PPPYPGESQTDLQPP

SPEN

2236

Q96T58
NPAPYPAPHLLQPGP

SP7

206

Q8TDD2
PPPVQPLPGTELEHY

ROBO2

1076

Q9HCK4
PPHDLAATQIPPAPP

TMEM209

116

Q96SK2
APLQPPSVPAPSDYP

ZMIZ2

731

Q8NF64
PAADYPTLPPPPLSQ

WASF2

371

Q9Y6W5
PEPPHSLPTHYQPEP

ZNF469

651

Q96JG9
YEIPPITPPNLPEPS

TOX2

76

Q96NM4
PPQPPPPDLSTELYY

ZNF462

1101

Q96JM2
HHIPSPPPAIPYELP

UBXN10

61

Q96LJ8
PELAPTAPLPYPAPE

VPS37B

181

Q9H9H4
VHRPGTPPPPYTVAP

WBP1

131

Q96G27
HRPEPLFIPPPPSYN

TRERF1

656

Q96PN7
PTHELPPYTPPPMLS

TRERF1

701

Q96PN7
PNLQPGYSPSPTHPP

THPO

286

P40225
PEEPPNYPAAPASDP

KDM5C

1321

P41229
KDQSPPPSPPPSYHP

KIAA1522

666

Q9P206
IYPLPDDPSVPAPPR

MYOF

1526

Q9NZM1